The Journal of Organic Chemistry · 2024 · 12 citations · 17 references
Natural SciencesChemistryMedicinal ChemistryOrganic ChemistryOrganic SynthesisIndole ChemistryIndole DerivativesIndole Synthesis
Herein, we present a sulfonylmethylation of indoles with aryl/alkyl hydrazides and sulfinates that provides viable access to sulfone compounds using rongalite as a C1 source. This protocol features readily available chemicals and simple operations, and the products were obtained in moderate to good yields.
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Rongalite as C1 Synthon in the Synthesis of Divergent Pyridines and Quinolines
Huan Gao, Liyun Zhou, Jie‐Ping Wan et al. · The Journal of Organic Chemistry · 2023 · 45 citations