A Metal‐Free Multicomponent Cascade Reaction for the Regiospecific Synthesis of 1,5‐Disubstituted 1,2,3‐Triazoles

Abstract

Alles an seinem Platz: Die Titelverbindungen werden regiospezifisch über eine Sequenz aus Michael-Addition, desacylierendem Diazotransfer und Cyclisierung synthetisiert. Mit dieser einfachen Methode, bei der drei kovalente Bindungen gebildet und zwei gespalten werden, lassen sich primäre Amine, einschließlich chiraler α-Amine herstellen. Ts=4-Toluolsulfonyl. As a service to our authors and readers, this journal provides supporting information supplied by the authors. Such materials are peer reviewed and may be re-organized for online delivery, but are not copy-edited or typeset. Technical support issues arising from supporting information (other than missing files) should be addressed to the authors. Please note: The publisher is not responsible for the content or functionality of any supporting information supplied by the authors. Any queries (other than missing content) should be directed to the corresponding author for the article.