Biomolecules · 2021 · 16 citations · 82 references
Life SciencesEntomologyMolecular BiologyEnzymologyInsect PathologyProtozoologyEnzyme InhibitionProtozoan Diseases Of InsectsNosema DiseaseNosema Infections In BeesPharmacological TherapyProtease Active SitesProtease InhibitionProteasome DysfunctionProteasome InhibitorsProteasome System
The microsporidia Nosema ceranae is an obligate intracellular parasite that causes honey bee mortality and contributes to colony collapse. Fumagillin is presently the only pharmacological control for N. ceranae infections in honey bees. Resistance is already emerging, and alternative controls are critically needed. Nosema spp. exhibit increased sensitivity to heat shock, a common proteotoxic stress. Thus, we hypothesized that targeting the Nosema proteasome, the major protease removing misfolded proteins, might be effective against N. ceranae infections in honey bees. Nosema genome analysis and molecular modeling revealed an unexpectedly compact proteasome apparently lacking multiple canonical subunits, but with highly conserved proteolytic active sites expected to be receptive to FDA-approved proteasome inhibitors. Indeed, N. ceranae were strikingly sensitive to pharmacological disruption of proteasome function at doses that were well tolerated by honey bees. Thus, proteasome inhibition is a novel candidate treatment strategy for microsporidia infection in honey bees.
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KEGG: Kyoto Encyclopedia of Genes and Genomes
Minoru Kanehisa · Nucleic Acids Research · 2000 · 39.2K citations · Full text
KEGG: Kyoto Encyclopedia of Genes and Genomes
Hiroyuki Ogata, Susumu Goto, Kazushige Sato et al. · Nucleic Acids Research · 1999 · 32.4K citations · Full text
Structure of 20S proteasome from yeast at 2.4Å resolution
M. Groll, Lars Ditzel, Jan Löwe et al. · Nature · 1997 · 2.3K citations
A gated channel into the proteasome core particle.
M. Groll, Michael H. Glickman, Daniel Finley et al. · Nature Structural Biology · 2000 · 808 citations