Concepedia

Rh(<scp>iii</scp>)-Catalyzed tandem C(sp<sup>2</sup>)–H allylation/<i>N</i>-alkylation annulation of arene amides with 2-alkylidenetrimethylene carbonates

Hui Xie, Jin-Yi Liang, Zhuojun Huang, Bing Shu, Yi‐Chuan Zheng, Yanzhi Liu, Shaoyong Chen, Xu‐Ge Liu, Shang‐Shi Zhang

Organic Chemistry Frontiers · 2021 · 25 citations · 35 references

DOI

Concepts

Abstract

A Rh( iii )-catalyzed tandem C(sp 2 )–H allylation/ N -alkylation annulation reaction of arene amides employing 5-methylene-1,3-dioxan-2-one as an efficient allyl source has been disclosed for the first time.

References

35

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