Concepedia

Palladium‐Catalyzed Oxidative Arylation of 1<i>H</i>‐Indazoles with Arenes

Khadija Gambouz, Abdelmoula El Abbouchi, Sarah Nassiri, Franck Suzenet, Mostapha Bousmina, Mohamed Akssira, Gérald Guillaumet, Saı̈d El Kazzouli

European Journal of Organic Chemistry · 2020 · 13 citations · 46 references

DOI

Concepts

Abstract

A simple method for the direct Pd(OAc) 2 ‐catalyzed oxidative arylation of inactivated 1 H ‐indazole derivatives with simple arenes is reported. This method exhibits good reaction efficiency and good functional‐group tolerance. Using the developed method, 28 arylated products were prepared in yields up to 80 %.

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