Inorganic Chemistry Frontiers · 2020 · 20 citations · 70 references
Natural SciencesChemistryMedicinal ChemistryBiophysical ChemistryDrug DesignStructure-activity RelationshipsAmyloid FormationChemical BondingChemical ReactionsCoordination ChemistryLigand BindingMetal-ligand BondingLigand Effects On ReactivityMetal Binding FeaturesMetal Ion Binding To Aggregation-prone ProteinsMetal-based TherapeuticsMetal-binding Properties
New examples of azamacrocyclic metal chelators that modulate the interactions between metal ions and Aβ and the reactivities of metal–Aβ were developed under criteria based on structural and functional variations on the backbone of<bold>Cyclam</bold>.
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