Concepedia

Pyridinium derivatives of 3-aminobenzenesulfonamide are nanomolar-potent inhibitors of tumor-expressed carbonic anhydrase isozymes CA IX and CA XII

Süleyman Akocak, Özlen Güzel-Akdemir, Rajesh Kishore Kumar Sanku, Samson S. Russom, Bogdan I. Iorga, Claudiu T. Supuran, Marc A. Ilies

Bioorganic Chemistry · 2020 · 36 citations · 56 references

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References

56

Improved protein–ligand docking using GOLD

Marcel L. Verdonk, Jason C. Cole, Michael J. Hartshorn et al. · Proteins Structure Function and Bioinformatics · 2003 · 3K citations · Full text

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The Carbon Dioxide Hydration Activity of Carbonic Anhydrase

Raja G. Khalifah · Journal of Biological Chemistry · 1971 · 1.9K citations · Full text

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Hypoxia-inducible expression of tumor-associated carbonic anhydrases.

Charles C. Wykoff, Nigel Beasley, Peter H. Watson et al. · PubMed · 2000 · 1.3K citations

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Hypoxia-Inducible Carbonic Anhydrase IX and XII Promote Tumor Cell Growth by Counteracting Acidosis through the Regulation of the Intracellular pH

Johanna Chiche, Karine Ilc, Julie Laferrière et al. · Cancer Research · 2008 · 746 citations

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Crystal structure of the catalytic domain of the tumor-associated human carbonic anhydrase IX

Vincenzo Alterio, Mika Hilvo, Anna Di Fiore et al. · Proceedings of the National Academy of Sciences · 2009 · 519 citations · Full text

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