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Exploring occupancy of the histamine H<sub>3</sub> receptor by pitolisant in humans using PET

DOIFull Paper Access

21

Citations

25

References

2020

Year

Pablo Rusjan, Pamela Sabioni, Patricia Di Ciano, Esmaeil Mansouri, Isabelle Boileau, Alexia Laveillé, Marc Capet, Thierry Duvauchelle, Jean‐Charles Schwartz, Philippe Robert,
British Journal of Pharmacology

Abstract

The administration of pitolisant (40 mg) produces a high occupancy of H<sub>3</sub> receptors and may be a new tool for the treatment of a variety of CNS disorders that are associated with mechanisms involving H<sub>3</sub> receptors.

References

YearCitations

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