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Coumarins from<i>Magydaris pastinacea</i>as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation

Benedetta Fois, Simona Distinto, Rita Meleddu, Serenella Deplano, Elias Maccioni, Costantino Floris, Antonella Rosa, Mariella Nieddu, Pierluigi Caboni, Claudia Sissi,

Journal of Enzyme Inhibition and Medicinal Chemistry · 2020 · 33 citations · 40 references

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Abstract

of 5.7 nM. The cytotoxicity of the most interesting compounds on HeLa cancer cells was also investigated.

References

40

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Macromodel—an integrated software system for modeling organic and bioorganic molecules using molecular mechanics

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The Carbon Dioxide Hydration Activity of Carbonic Anhydrase

Raja G. Khalifah · Journal of Biological Chemistry · 1971 · 1.9K citations · Full text

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