Transition-metal-free lactamization of C(sp<sup>3</sup>)–H bonds with CO<sub>2</sub>: facile generation of pyrido[1,2-<i>a</i>]pyrimidin-4-ones

Zhen Zhang, Xiaoyu Zhou, Jin‐Gui Wu, Lei Song, Da‐Gang Yu

Green Chemistry · 2019 · 38 citations · 53 references

Concepts

Abstract

A novel carbonylation of C(sp<sup>3</sup>)–H bonds in pyridylamines with one atmosphere of CO<sub>2</sub> is reported to synthesize important pyrimidinones in good yields.

References

53