Concepedia

Dual-target inhibitors of mycobacterial aminoacyl-tRNA synthetases among <i>N</i>-benzylidene-<i>N</i>′-thiazol-2-yl-hydrazines

O. P. Kovalenko, Galyna P. Volynets, Mariia Yu. Rybak, Sergiy A. Starosyla, O. I. Gudzera, Volodymyr G. Bdzhola, S. M. Yarmoluk, Helena I. Boshoff, M. A. Tukalo

MedChemComm · 2019 · 27 citations · 25 references

DOIFull text

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Concepts

Abstract

A screen of 37 compounds identified four inhibitors that exhibited dual on-target activity against <italic>Mycobacterium tuberculosis</italic> aminoacyl-tRNA synthetases.

References

25

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