Publication | Closed Access
Exploring oxidovanadium(<scp>iv</scp>) homoleptic complexes with 8-hydroxyquinoline derivatives as prospective antitrypanosomal agents
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Citations
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References
2019
Year
8-Hydroxyquinoline Derivatives LAntiparasitic AgentHeterocycle ChemistryChemical BiologyPharmaceutical ChemistryParasite GenomicsHomoleptic ComplexesMedicinal ChemistryHigh SelectivitiesToxicologyProspective Antitrypanosomal Agents8-Hydroxyquinoline DerivativesDerivativesBiochemistryParasitic ProtozoaPharmacologyNatural SciencesMedicineDrug Discovery
[V<sup>IV</sup>O(L-H)<sub>2</sub>] and [V<sup>V</sup>O(OCH<sub>3</sub>)(L-H)<sub>2</sub>] compounds of 8-hydroxyquinoline derivatives L showed activity against<italic>Trypanosoma cruzi</italic>and<italic>Leishmania infantum</italic>and high selectivities. Metallomics and interaction with BSA, apo-HTF and DNA were studied.
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