Concepedia

ASYMMETRIC SYNTHESIS OF 1-AMINOALKYLPHOSPHONIC ACIDS

Robert Jacquier, Mohamed Lhassani, C. PETRUS, FRANCOISE PETRUS

Phosphorus, sulfur, and silicon and the related elements · 1993 · 17 citations · 7 references

DOI

Concepts

Abstract

Abstract Asymmetric synthesis of Phe and Tyr phosphonic analogous has been achieved by diastereoselective alkylation of chiral 1,2,3-oxazaphospholanes, the latter being readily obtained from (-) ephedrine and chloromethylphosphonic dichloride.

References

7

OPTICALLY ACTIVE 1-AMINOALKYLPHOSPHONIC ACIDS

Balram Dhawan, Derek Redmore · Phosphorous and Sulfur and the Related Elements · 1987 · 178 citations

, , +15

A versatile asymmetric synthesis of α-amino α-alkyl-phosphonic acids of high enantiomeric purity

Stephen Hanessian, Youssef L. Bennani · Tetrahedron Letters · 1990 · 100 citations

, , +8

1,3,2-Oxazaphospholidines from (–)-ephedrine. Intermediates for the stereospecific synthesis of optically active dialkyl alkylphosphonothioates and -selenoates, trialkyl phosphoro-thioates and -selenoates, dialkyl methylphosphonates, and trialkyl phosphates

David B. Cooper, C. Richard Hall, J. M. Harrison et al. · Journal of the Chemical Society Perkin Transactions 1 · 1977 · 86 citations

, , +9

Asymmetric electrophilic amination of chiral phosphorus-stabilized anions

Scott E. Denmark, Naoto Chatani, Sunil V. Pansare · Tetrahedron · 1992 · 82 citations

, , +7

Peptides Containing Aminophosphonic Acids. II. The Synthesis of Tripeptide Analogs

Kiyoshi Yamauchi, Masayoshi Kinoshita, Minoru Imoto · Bulletin of the Chemical Society of Japan · 1972 · 33 citations

, , +9