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The Intramolecular Azide Cycloaddition Route to Triazolam Analogues
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1995
Year
Key StepPharmaceutical ChemistryHeterocyclicMedicineFacile SynthesisIsatoic AnhydridesOrganic ChemistryClick ChemistryHeterocycle ChemistryPharmacologyTriazolam AnaloguesDrug Discovery
A facile synthesis of [1,2,3]triazolo[1,5-a]benzodiazepines starting from isatoic anhydrides and involving an intramolecular azide cycloaddition as the key step is reported.