Concepedia

Synthesis of novel pyrrolidin‐2‐ones: γ‐aminobutyric acid cyclic analogues

Sahar Al Akoum Ebrik, Benoı̂t Rigo, Claude Vaccher, M.‐P. VACCHER, Nathalie Flouquet, Michel Debaert, Pascal Berthelot

Journal of Heterocyclic Chemistry · 1998 · 13 citations · 19 references

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Abstract

Abstract Some new N ‐substituted pyrrolidin‐2‐ones, cyclic analogues of baclofen and of 3‐(5‐methoxybenzo‐[ b ]furan‐2‐yl)‐γ‐aminobutyric acid, have been prepared and characterized, starting from 4‐(4‐chlorophenyl)‐pyrrolidin‐2‐one and 4‐(5‐methoxybenzo[ b ]furan‐2‐yl)pyrrolidin‐2‐one.

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