Stereochemistry of phase-1 metabolites of mephedrone determines their effectiveness as releasers at the serotonin transporter

Pharmacological characterization of designer cathinones<i>in vitro</i>

TA Buser, Massimiliano Donzelli, York Schramm et al. · British Journal of Pharmacology · 2012 · 673 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +9

The molecular mechanism of "ecstasy" [3,4-methylenedioxy-methamphetamine (MDMA)]: serotonin transporters are targets for MDMA-induced serotonin release.

Gary Rudnick, S C Wall · Proceedings of the National Academy of Sciences · 1992 · 533 citations

Medicine, Biochemistry, Pharmacology +17

Clinical experience with and analytical confirmation of “bath salts” and “legal highs” (synthetic cathinones) in the United States

Henry A. Spiller, Mark L. Ryan, Robert G. Weston et al. · Clinical Toxicology · 2011 · 525 citations

Pharmacy, Clinical Toxicology, Toxicology +15

The Designer Methcathinone Analogs, Mephedrone and Methylone, are Substrates for Monoamine Transporters in Brain Tissue

Michael H. Baumann, Mario Ayestas, John S. Partilla et al. · Neuropsychopharmacology · 2011 · 438 citations

Medicine, Neuroscience, Pharmacology +16

Receptor interaction profiles of novel psychoactive tryptamines compared with classic hallucinogens

Anna Rickli, Olivier D. Moning, Marius C. Hoener et al. · European Neuropsychopharmacology · 2016 · 371 citations

Medicine, Medicinal Chemistry, Pharmacology +12