Concepedia

A cascade synthesis, in vitro cholinesterases inhibitory activity and docking studies of novel Tacrine-pyranopyrazole derivatives

Chamseddine Derabli, Imen Boualia, Ahmed B. Abdelwahab, Raouf Boulcina, Gilbert Kirsch, Abdelmadjid Debache

Bioorganic & Medicinal Chemistry Letters · 2018 · 60 citations · 29 references

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References

29

AutoDock Vina: Improving the speed and accuracy of docking with a new scoring function, efficient optimization, and multithreading

Oleg Trott, Arthur J. Olson · Journal of Computational Chemistry · 2009 · 37.1K citations · Full text

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A new and rapid colorimetric determination of acetylcholinesterase activity

George L. Ellman, K. Diane Courtney, Valentino Andres et al. · Biochemical Pharmacology · 1961 · 26.9K citations

, , +14

Structure-based discovery of an organic compound that binds Bcl-2 protein and induces apoptosis of tumor cells

Jialun Wang, Dongxiang Liu, Zhijia Zhang et al. · Proceedings of the National Academy of Sciences · 2000 · 1.2K citations

, , +17

Hepatotoxic Effects of Tacrine Administration in Patients With Alzheimer's Disease

Paul B. Watkins · JAMA · 1994 · 787 citations

, , +17

Identification of chemically diverse Chk1 inhibitors by receptor-based virtual screening

Nicolas Foloppe, Lisa M. Fisher, Rob Howes et al. · Bioorganic & Medicinal Chemistry · 2006 · 363 citations · Full text

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