Gold‐Catalyzed Intermolecular [4+2] Annulation of 2‐Ethynylanilines with Ynamides: An Access to Substituted 2‐Aminoquinolines

Abstract

Abstract A gold‐catalyzed intermolecular [4+2] annulation of easily accessible 2‐ethynylanilines with ynamides offers a highly region‐selective, modular, efficient, and atom‐economical strategy for the synthesis of substituted 2‐aminoquinolines in up to 93% yield. magnified image