Metal-catalyzed privileged 2- and 3-functionalized indole synthesis*

Synthesis of 2,3-Disubstituted Indoles via Palladium-Catalyzed Annulation of Internal Alkynes

Richard C. Larock, Mitchell D. Refvik · The Journal of Organic Chemistry · 1998 · 598 citations

Natural Sciences, Chemistry, Medicinal Chemistry +13

Rhodium(III)-Catalyzed Indole Synthesis Using N–N Bond as an Internal Oxidant

Baoqing Liu, Chao Song, Chao Sun et al. · Journal of the American Chemical Society · 2013 · 343 citations

Natural Sciences, Chemistry, Medicinal Chemistry +17

Palladium-Catalyzed Aerobic Oxidative Cyclization of <i>N</i>-Aryl Imines: Indole Synthesis from Anilines and Ketones

Ye Wei, Indubhusan Deb, Naohiko Yoshikai · Journal of the American Chemical Society · 2012 · 340 citations

Natural Sciences, Chemistry, Medicinal Chemistry +14

A Palladium-Catalyzed Method for the Preparation of Indoles via the Fischer Indole Synthesis

Seble Wagaw, Bryant H. Yang, Stephen L. Buchwald · Journal of the American Chemical Society · 1999 · 277 citations

Natural Sciences, Chemistry, Medicinal Chemistry +12

Development of an Efficient Procedure for Indole Ring Synthesis from 2-Ethynylaniline Derivatives Catalyzed by Cu(II) Salts and Its Application to Natural Product Synthesis

Kou Hiroya, Shin Itoh, Takao Sakamoto · The Journal of Organic Chemistry · 2004 · 261 citations

Natural Sciences, Chemistry, Medicinal Chemistry +15