Concepedia

3H-pyrazolo[4,3-f]quinoline haspin kinase inhibitors and anticancer properties

Clement Opoku‐Temeng, Neetu Dayal, Moloud Aflaki Sooreshjani, Herman O. Sintim

Bioorganic Chemistry · 2018 · 41 citations · 14 references

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Open access

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References

14

The kinase haspin is required for mitotic histone H3 Thr 3 phosphorylation and normal metaphase chromosome alignment

Jun Dai, Sammy Sultan, Stephen S. Taylor et al. · Genes & Development · 2005 · 375 citations · Full text

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On the Mechanism of the Skraup−Doebner−Von Miller Quinoline Synthesis

Scott E. Denmark, Srikanth Venkatraman · The Journal of Organic Chemistry · 2006 · 210 citations

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Structure and functional characterization of the atypical human kinase haspin

Jeyanthy Eswaran, Debasis Patnaik, P. Filippakopoulos et al. · Proceedings of the National Academy of Sciences · 2009 · 192 citations · Full text

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Antitumor activity of a small-molecule inhibitor of the histone kinase Haspin

Dori Huertas, Marta Soler, Jemina Moretó et al. · Oncogene · 2011 · 121 citations · Full text

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A small-molecule inhibitor of Haspin alters the kinetochore functions of Aurora B

Anna De Antoni, Stefano Maffini, Stefan Knapp et al. · The Journal of Cell Biology · 2012 · 115 citations · Full text

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