Journal of Enzyme Inhibition and Medicinal Chemistry · 2017 · 12 citations · 32 references
PharmacyMedicinal ChemistryPharmacologyDrug DesignDrug DiscoveryStructure-activity RelationshipsLead Compound DesignLigand BindingMolecular DockingProtein-ligand DockingReceptor PharmacologyStructure-activity Relationship AnalysisAdenosine Receptor ModulationAdenosine Receptor SignalingBenzoxazole SynthesisChemical Synthesis Of AnaloguesDocking-based Drug DesignDrug Receptor PharmacologyMedicinal Chemistry ApplicationsStructure-based Ligand Design
= 10 μm), can be easily modulated and thus considered as relevant starting points for further hit-to-lead optimisation.
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Structural Basis for Allosteric Regulation of GPCRs by Sodium Ions
Wei Liu, Eugene Chun, Aaron A. Thompson et al. · Science · 2012 · 965 citations · Full text