Iodine-catalyzed C3-formylation of indoles using hexamethylenetetramine and air

Direct and Practical Synthesis of 2-Arylbenzoxazoles Promoted by Activated Carbon

Yuka Kawashita, Natsuki Nakamichi, Hirotoshi Kawabata et al. · Organic Letters · 2003 · 225 citations

Natural Sciences, Chemistry, Catalysis +10

Mild and Selective Ru-Catalyzed Formylation and Fe-Catalyzed Acylation of Free (N–H) Indoles Using Anilines as the Carbonyl Source

Wenliang Wu, Weiping Su · Journal of the American Chemical Society · 2011 · 212 citations

Natural Sciences, Chemistry, Catalysis +14

Fluorination of 3-(3-(Piperidin-1-yl)propyl)indoles and 3-(3-(Piperazin-1-yl)propyl)indoles Gives Selective Human 5-HT_1D Receptor Ligands with Improved Pharmacokinetic Profiles

Monique B. van Niel, Ian Collins, Margaret S. Beer et al. · Journal of Medicinal Chemistry · 1999 · 157 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +16

Aerobic Transition-Metal-Free Visible-Light Photoredox Indole C-3 Formylation Reaction

Xiang Li, Xiangyong Gu, Yongjuan Li et al. · ACS Catalysis · 2014 · 154 citations

Natural Sciences, Biochemistry, Chemistry +13

Cu(ii)-catalyzed C–H (SP3) oxidation and C–N cleavage: base-switched methylenation and formylation using tetramethylethylenediamine as a carbon source

Lei Zhang, Peng Chen, Dan Zhao et al. · Chemical Communications · 2012 · 118 citations

Natural Sciences, Chemistry, Catalysis +16