Journal of Heterocyclic Chemistry · 2017 · 20 citations · 23 references
MedicineCardiologyPharmacologyCardiovascular PharmacotherapyDrug DesignSynthetic Medicinal ChemistryCardiac Ion ChannelsCardiac MedicationsCardiac PharmacotherapyCardiovascular PharmacodynamicsIon Channel PharmacologyIon Channel PhysiologyCalcium Channel PharmacologyCalcium Channel PhysiologyL-type Calcium CurrentOverviewVoltage-gated Calcium Channels
The data on historical development and modern design approaches for calcium channels blockers (mainly L‐type) are summarized in this review. Chemical groups such as dihydropyridine and hydropyrimidine derivatives, as well as phenylalkylamines and benzothiazepines are discussed.
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Comprehensive Medicinal Chemistry
Quantitative Structure-Activity Relationships · 1991 · 749 citations
George C. Rovnyak, S. David Kimball, Barbara Beyer et al. · Journal of Medicinal Chemistry · 1995 · 549 citations · Full text
Hantzsch-type dihydropyridine hypotensive agents
Bernard Loev, M. M. GOODMAN, Kenneth M. Snader et al. · Journal of Medicinal Chemistry · 1974 · 346 citations