Organic Letters · 2017 · 45 citations · 34 references
PharmacyMedicinal ChemistryPharmaceuticsDrug DeliveryDrug DesignDrug DiscoveryControlled Release ProdrugsProdrug Activation MechanismsProdrug Release Mechanisms
Employing an intramolecular cycloaddition reaction, we have developed a series of SO 2 prodrugs with tunable release rates with half-lives ranging from minutes to days.
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