Concepedia

Transition-metal free direct difluoromethylthiolation of electron-rich aromatics with difluoromethanesulfonyl chloride

Xia Zhao, Aoqi Wei, Tianjiao Li, Zhiyang Su, Jun Chen, Kui Lu

Organic Chemistry Frontiers · 2016 · 42 citations · 34 references

DOI

Concepts

Abstract

A new method for phosphine-mediated difluoromethylthiolation of indoles and other electron-rich aromatics using difluoromethanesulfonyl chloride was developed.

References

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