Concepedia
Medicinal Chemistry Research · 2010 · 21 citations · 28 references
PharmacyChemistryMedicinal ChemistryDrug DiscoveryOrganic ChemistryStructure-activity RelationshipsEnzyme InhibitionUrease ActivityUrease InhibitorsUrease Test
28
Phenol-hypochlorite reaction for determination of ammonia
Muriel W. Weatherburn · Analytical Chemistry · 1967 · 4.1K citations
Natural Sciences, Chemistry, Analytical Chemistry +5
Fast Calculation of Molecular Polar Surface Area as a Sum of Fragment-Based Contributions and Its Application to the Prediction of Drug Transport Properties
Peter Ertl, Bernhard Rohde, Paul M. Selzer · Journal of Medicinal Chemistry · 2000 · 3K citations
Pharmacy, Chemistry, Pharmacology +15
Synthesis and antitubercular activity of imidazo[2,1-b]thiazoles
Aldo Andreani, Massimiliano Granaiola, Alberto Leoni et al. · European Journal of Medicinal Chemistry · 2001 · 165 citations
Pharmacy, Medicinal Chemistry, Pharmacology +9
A class of selective antibacterials derived from a protein kinase inhibitor pharmacophore
J. Richard Miller, Steve Dunham, Igor Mochalkin et al. · Proceedings of the National Academy of Sciences · 2009 · 160 citations · Full text
Pharmacy, Medicinal Chemistry, Pharmacology +17
Synthesis and biological evaluation of imidazo[1,2-a]pyridine derivatives as novel PI3 kinase p110α inhibitors
Masahiko Hayakawa, Hiroyuki Kaizawa, Kenichi Kawaguchi et al. · Bioorganic & Medicinal Chemistry · 2006 · 124 citations · Full text
Pharmacy, Medicinal Chemistry, Pharmacology +10