Concepedia

Abstract

SUMMARY Antibiotics and vehicles used in the treatment and prevention of mastitis were tested in vitro to determine effects on phagocytosis of 32 P-labeled Staphylococcus aureus ([ 32 P] sa ) by bovine polymorphonuclear leukocytes ( pmn ) isolated from milk. Ampicillin, lincomycin, erythromycin, tetracycline, neomycin, penicillin G, streptomycin, cephalothin, nitrofurantoin, gentamicin, dicloxacillin, rifampin, trimethoprim, amikacin, novobiocin-penicillin, polymyxin B, and tiamulin were tested at in vitro concentrations of 1,000, 500, and 10 μg/ml, and sulfamethoxazole and chloramphenicol at 4,000, 2,000, and 10 μg/ml of incubation mixture. These dilutions were equivalent to antibiotic values in milk at 0, 6, and 12 hours after injection into the mammary gland. Vehicles included peanut oil, mineral oil, 3% cabosil in peanut oil, 2% aluminum monostearate in peanut oil, 25% polyethylene glycol ( peg ) in an aqueous base, 25% peg in mineral oil, and 25% peg in peanut oil. These were tested at dilutions of 1:100, 1:1,000, 1:5,000, and 1:10,000. The percentage of phagocytosis was determined and was compared with the percentage of phagocytosis in phosphate-buffered saline solution ( pbss ). Antibiotics and vehicles were diluted in 0.0132 M pbss (pH 7.4); combined with skimmed milk, pmn (12.5 × 10 6 ), and [ 32 P] sa (50 × 10 6 ); and incubated for 1 hour (37 C, no rocking) followed by rocking for 1 hour. A minimum of 2 runs for the antibiotics and 3 runs for the vehicles were performed with all concentrations or dilutions assayed in a single day's run. Phagocytosis was significantly ( P < 0.05) reduced at the high and intermediate concentrations for tiamulin, nitrofurantoin, rifampin, chloramphenicol, and amikacin, and at the high concentrations for gentamicin, tetracycline, and novobiocin-penicillin. The only vehicle that inhibited phagocytosis significantly was peanut oil without additives at the 1:100 dilution.