Gold‐Catalyzed Aminoalkenylation of β‐Amino‐1,<i>n</i>‐Diynols to Cycloalkyl‐, Piperidinyl‐ and Pyranyl‐Fused Pyrroles

Prasath Kothandaraman, Yichao Zhao, BoRa Lee, Clarrisa Jia Le Ng, Jun Yi Lee, Benjamin James Ayers, Philip Wai Hong Chan

Advanced Synthesis & Catalysis · 2016 · 21 citations · 74 references

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Abstract

Abstract A synthetic method to prepare cycloalkyl‐, piperidinyl‐ and pyranyl‐fused pyrroles efficiently by gold(I)‐catalyzed dehydrative aminoalkenylation of β‐amino‐1, n ‐diynols under mild conditions at room temperature is described. magnified image

References

74