Organic Process Research & Development · 2014 · 23 citations · 16 references
PharmacyChemistryMedicinal ChemistryDrug DiscoveryOrganic ChemistrySynthetic Medicinal ChemistryEnzyme InhibitionFibrin FormationAntifibrinolytic AgentsEnzymatic ResolutionIsoxazole ChemistryIsoxazole SynthesisNegishi Coupling
A practical and chromatography-free multikilogram synthesis of a 3-isoxazolol containing antifibrinolytic agent, AZD6564, has been developed in eight steps and 7% overall yield starting from methyl 2-chloroisonicotinate. Highlights in the synthesis are a Negishi coupling and an enzymatic resolution of a racemic ester.
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Iron-Catalyzed Cross-Coupling Reactions
Alois Fürstner, Andreas Leitner, Marı́a Méndez et al. · Journal of the American Chemical Society · 2002 · 820 citations
Chaoyang Dai, Gregory C. Fu · Journal of the American Chemical Society · 2001 · 399 citations
Efficient Asymmetric Hydrogenation of Pyridines
Frank Glorius, Nick Spielkamp, S. Holle et al. · Angewandte Chemie International Edition · 2004 · 222 citations