Concepedia

Cardanol-derived AChE inhibitors: Towards the development of dual binding derivatives for Alzheimer's disease

Laís Flávia Nunes Lemes, Giselle de Andrade Ramos, Andressa Souza de Oliveira, Fernanda Motta R. da Silva, Gina C. Couto, Marina da Silva Boni, Marcos Jorge R. Guimarães, Isis Nem de Oliveira Souza, Manuela Bartolini, Vincenza Andrisano,

European Journal of Medicinal Chemistry · 2015 · 92 citations · 35 references

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35

A new and rapid colorimetric determination of acetylcholinesterase activity

George L. Ellman, K. Diane Courtney, Valentino Andres et al. · Biochemical Pharmacology · 1961 · 26.9K citations

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Molecular Properties That Influence the Oral Bioavailability of Drug Candidates

Daniel F. Veber, Stephen R. Johnson, Hung‐Yuan Cheng et al. · Journal of Medicinal Chemistry · 2002 · 8.1K citations

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Improved protein–ligand docking using GOLD

Marcel L. Verdonk, Jason C. Cole, Michael J. Hartshorn et al. · Proteins Structure Function and Bioinformatics · 2003 · 3K citations · Full text

, , +17

Fast Calculation of Molecular Polar Surface Area as a Sum of Fragment-Based Contributions and Its Application to the Prediction of Drug Transport Properties

Peter Ertl, Bernhard Rohde, Paul M. Selzer · Journal of Medicinal Chemistry · 2000 · 3K citations

, , +15

Alzheimer’s disease drug-development pipeline: few candidates, frequent failures

Jeffrey L. Cummings, Travis Morstorf, Kate Zhong · Alzheimer s Research & Therapy · 2014 · 1.7K citations · Full text

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