Concepedia

Orally active ghrelin receptor inverse agonists and their actions on a rat obesity model

Bitoku Takahashi, Hideaki Funami, Takehiko Iwaki, Hiroshi Maruoka, Makoto Shibata, Makoto Koyama, Asako Nagahira, Yoshiyuki Kamiide, Satomi Kanki, Yoshiyuki Igawa,

Bioorganic & Medicinal Chemistry · 2015 · 14 citations · 16 references

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16

Ghrelin is a growth-hormone-releasing acylated peptide from stomach

Masayasu Kojima, Hiroshi Hosoda, Yukari Date et al. · Nature · 1999 · 8.5K citations

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Ghrelin induces adiposity in rodents

Matthias H. Tschöp, David L. Smiley, Mark L. Heiman · Nature · 2000 · 3.9K citations

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The role of the gastric afferent vagal nerve in ghrelin-induced feeding and growth hormone secretion in rats

Yukari Date, Noboru Murakami, Koji Toshinai et al. · Gastroenterology · 2002 · 1.1K citations · Full text

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High Constitutive Signaling of the Ghrelin Receptor—Identification of a Potent Inverse Agonist

Birgitte Holst, Adam I. Cygankiewicz, Tine H. Jensen et al. · Molecular Endocrinology · 2003 · 516 citations

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Ghrelin Does Not Stimulate Food Intake in Patients with Surgical Procedures Involving Vagotomy

Carel W. le Roux, Nicola M. Neary, Tim Halsey et al. · The Journal of Clinical Endocrinology & Metabolism · 2005 · 264 citations · Full text

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