Three-component coupling of alkynes, Baylis–Hillman adducts and sodium azide: a new synthesis of substituted triazoles

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A Stepwise Huisgen Cycloaddition Process: Copper(I)-Catalyzed Regioselective “Ligation” of Azides and Terminal Alkynes

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Click Chemistry: Diverse Chemical Function from a Few Good Reactions

Hartmuth C. Kolb, M. G. Finn, K. Barry Sharpless · Angewandte Chemie International Edition · 2001 · 9.3K citations · Full text

Multicomponent Reactions with Isocyanides

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High-throughput Function Determination, Biomolecular Tool, Dna Microarrays +19