Concepedia

Novel heterocyclic glucocorticoids: in vitro profile and in vivo efficacy

Christopher F. Thompson, Christopher F. Thompson, Nazia Quraishi, Amjad Ali, James R. Tata, Milton L. Hammond, James M. Balkovec, Monica Einstein, Lan Ge, Georgianna Harris,

Bioorganic & Medicinal Chemistry Letters · 2005 · 45 citations · 16 references

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16

Goodman and Gilman's the Pharmacological Basis of Therapeutics

William H. Stigelman, D Pharm · Military Medicine · 1986 · 6.8K citations

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Dissociation of transactivation from transrepression by a selective glucocorticoid receptor agonist leads to separation of therapeutic effects from side effects

Heike Schäcke, Arndt Schottelius, Wolf‐Dietrich Döcke et al. · Proceedings of the National Academy of Sciences · 2003 · 470 citations · Full text

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Repression of inflammatory responses in the absence of DNA binding by the glucocorticoid receptor

Holger M. Reichardt · The EMBO Journal · 2001 · 429 citations · Full text

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Glucocorticoids inhibit the production of IL 6 from monocytes, endothelial cells and fibroblasts

Anders Waage, Geir Slupphaug, Refaat Shalaby · European Journal of Immunology · 1990 · 235 citations

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A Novel Antiinflammatory Maintains Glucocorticoid Efficacy with Reduced Side Effects

Michael J. Coghlan, Peer B. Jacobson, Ben Lane et al. · Molecular Endocrinology · 2003 · 221 citations

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