Concepedia

Synthesis and biological evaluation of γ-aminophosphonates as potent, subtype-selective sphingosine 1-phosphate receptor agonists and antagonists

Frank W. Foss, Ashley H. Snyder, Michael D. Davis, Michael Rouse, Mark D. Okusa, Kevin R. Lynch, Timothy L. Macdonald

Bioorganic & Medicinal Chemistry · 2006 · 158 citations · 33 references

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References

33

Lymphocyte egress from thymus and peripheral lymphoid organs is dependent on S1P receptor 1

Mehrdad Matloubian, Charles G. Lo, Guy Cinamon et al. · Nature · 2004 · 2.5K citations

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A greatly improved procedure for ruthenium tetroxide catalyzed oxidations of organic compounds

Per H. J. Carlsen, Tsutomu Katsuki, Victor S. Martı́n et al. · The Journal of Organic Chemistry · 1981 · 1.6K citations

, , +7

PyBOP®: A new peptide coupling reagent devoid of toxic by-product

J. H. Coste, Dung Le‐Nguyen, B. CASTRO · Tetrahedron Letters · 1990 · 614 citations

, , +7

Enhancement of capillary leakage and restoration of lymphocyte egress by a chiral S1P1 antagonist in vivo

Marta Sanna, Sheng‐Kai Wang, Pedro J. Gonzalez‐Cabrera et al. · Nature Chemical Biology · 2006 · 401 citations · Full text

, , +16

Sphingosine 1-Phosphate Analogs as Receptor Antagonists

Michael D. Davis, Jeremy J. Clemens, Timothy L. Macdonald et al. · Journal of Biological Chemistry · 2004 · 270 citations · Full text

, , +17