Biochemical and Biophysical Research Communications · 1985 · 31 citations · 6 references
PharmacyMedicinal ChemistryPharmacologyDrug DesignDrug DiscoveryEnzymologyAmino Acid ChemistryEnzyme DesignEnzyme InhibitionPeptide ChemistryPeptide Drug DiscoveryPeptidomimetic DesignAngiotensin-converting Enzyme Inhibitory PeptidesPeptide Analogue DesignPeptide Drug DevelopmentPeptide Medicinal ChemistryTransition-state Analogue Inhibitors
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A new class of angiotensin-converting enzyme inhibitors
Arthur A. Patchett, Elbert E. Harris, Edward W. Tristram et al. · Nature · 1980 · 706 citations
Enzymatic Catalysis and Transition-State Theory
Gustav E. Lienhard · Science · 1973 · 509 citations
Suicide substrates: mechanism-based enzyme inactivators
Christopher T. Walsh · Tetrahedron · 1982 · 443 citations