Publication | Closed Access
Naphthoquinone-based chalcone hybrids and derivatives: synthesis and potent activity against cancer cell lines
47
Citations
37
References
2014
Year
Medicinal ChemistryDiversity Oriented SynthesisDerivativesCancer Cell LinesMedicineNaphthoquinone-based Chalcone HybridsOrganic ChemistryImmunotherapeuticsPotent ActivityAnti-cancer AgentPromising Anticancer ActivityCytotoxic ActivityPharmacologyRadiation OncologyPharmaceutical ChemistryDrug Discovery
Naphthoquinone-based chalcone hybrids were synthesized and evaluated for their cytotoxic activity against four cancer cell lines and PBMC. Some of the hybrids exhibited promising anticancer activity with IC<sub>50</sub> values < 1 μM.
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