Concepedia

Azide‐Free Synthesis of 1,2,3‐Triazoles: New Opportunity for Sustainable Synthesis

Jie‐Ping Wan, Deqing Hu, Yunyun Liu, Shou‐Ri Sheng

ChemCatChem · 2015 · 44 citations · 49 references

DOI

Concepts

Abstract

A bright future for triazoles: The recent breakthrough in the synthesis of 1,2,3-triazoles is highlighted for its significance as a new tool in the chemistry of 1,2,3-triazoles following the classical CuAAC and metal-free protocols.

References

49

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Peptidotriazoles on Solid Phase:  [1,2,3]-Triazoles by Regiospecific Copper(I)-Catalyzed 1,3-Dipolar Cycloadditions of Terminal Alkynes to Azides

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A Strain-Promoted [3 + 2] Azide−Alkyne Cycloaddition for Covalent Modification of Biomolecules in Living Systems

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1,3‐Dipolar Cycloadditions. Past and Future

Rolf Huisgen · Angewandte Chemie International Edition in English · 1963 · 2.8K citations

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Kinetics and Mechanism of 1,3‐Dipolar Cycloadditions

Rolf Huisgen · Angewandte Chemie International Edition in English · 1963 · 1.2K citations

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