Concepedia

Chemical modification of epibatidine causes a switch from agonist to antagonist and modifies its selectivity for neuronal nicotinic acetylcholine receptors

Jörg E Spang, Sonia Bertrand, G. Westera, J. T. Patt, P. August Schubiger, Daniel Bertrand

Chemistry & Biology · 2000 · 39 citations · 41 references

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41

On the nature of allosteric transitions: A plausible model

Jacques Monod, Jeffries Wyman, Jean‐Pierre Changeux · Journal of Molecular Biology · 1965 · 8.9K citations

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Molecular cloning, functional properties, and distribution of rat brain alpha 7: a nicotinic cation channel highly permeable to calcium

Philippe Séguéla, Jacques I. Wadiche, Kelly Dineley‐Miller et al. · Journal of Neuroscience · 1993 · 1.5K citations · Full text

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Mutations in the channel domain alter desensitization of a neuronal nicotinic receptor

Frédéric Revah, Daniel Bertrand, Jean‐Luc Galzi et al. · Nature · 1991 · 525 citations

, , +14

Choline is a Selective Agonist of α7 Nicotinic Acetylcholine Receptors in the Rat Brain Neurons

Manickavasagom Alkondon, Edna F. R. Pereira, Wellington S. Cartes et al. · European Journal of Neuroscience · 1997 · 441 citations

, , +17

Epibatidine, a potent analgetic and nicotinic agonist.

Barbara Badio, John W. Daly · Molecular Pharmacology · 1994 · 387 citations

, , +12