Structure–activity relationships of 2-aryl-1H-indole inhibitors of the NorA efflux pump in Staphylococcus aureus

Efflux-mediated fluoroquinolone resistance in Staphylococcus aureus

Glenn W. Kaatz, S M Seo, C. A. Ruble · Antimicrobial Agents and Chemotherapy · 1993 · 412 citations

Life Sciences, Molecular Biology, Pharmacology +17

Direct C-Arylation of Free (NH)-Indoles and Pyrroles Catalyzed by Ar−Rh(III) Complexes Assembled In Situ

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Natural Sciences, Chemistry, Catalysis +16

Multiple Novel Inhibitors of the NorA Multidrug Transporter of <i>Staphylococcus aureus</i>

Penelope N. Markham, Eric Westhaus, Katya Klyachko et al. · Antimicrobial Agents and Chemotherapy · 1999 · 217 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13

Flavonolignan and Flavone Inhibitors of a <i>Staphylococcus </i><i>a</i><i>ureus</i> Multidrug Resistance Pump:  Structure−Activity Relationships

Nathan R. Guz, Frank R. Stermitz, Jeffrey B. Johnson et al. · Journal of Medicinal Chemistry · 2000 · 153 citations

Pharmacy, Medicinal Chemistry, Pharmacology +16

Synthesis of functionalised 2-aryl-5-nitro-1H-indoles and their activity as bacterial NorA efflux pump inhibitors

Siritron Samosorn, John B. Bremner, Anthony R. Ball et al. · Bioorganic & Medicinal Chemistry · 2005 · 136 citations

Pharmacy, Chemistry, Medicinal Chemistry +10