Concepedia

7-Azaindole-3-acetic acid derivatives: Potent and selective CRTh2 receptor antagonists

David A. Sandham, Claire Adcock, Kamlesh Bala, Lucy Barker, Zarin Brown, Gerald Dubois, David C. Budd, Brian J. Cox, Robin A. Fairhurst, Markus Furegati,

Bioorganic & Medicinal Chemistry Letters · 2009 · 44 citations · 15 references

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References

15

Release of Prostaglandin D<sub>2</sub>into Human Airways during Acute Antigen Challenge

John Murray, André Bernard Tonnel, Alan Brash et al. · New England Journal of Medicine · 1986 · 475 citations

, , +14

Utilization of operational schemes for analog synthesis in drug design

John G. Topliss · Journal of Medicinal Chemistry · 1972 · 459 citations

, , +5

Fast Gradient HPLC Method to Determine Compounds Binding to Human Serum Albumin. Relationships with Octanol/Water and Immobilized Artificial Membrane Lipophilicity

Klára Valkó, Shenaz Nunhuck, Chris Bevan et al. · Journal of Pharmaceutical Sciences · 2003 · 331 citations

, , +12

Defining optimum lipophilicity and molecular weight ranges for drug candidates—Molecular weight dependent lower logD limits based on permeability

Michael J. Waring · Bioorganic & Medicinal Chemistry Letters · 2009 · 324 citations

, , +16

Molecular pharmacology of the human prostaglandin D<sub>2</sub> receptor, CRTH2

Nicole Sawyer, Elizabeth Cauchon, Anne Châteauneuf et al. · British Journal of Pharmacology · 2002 · 190 citations · Full text

, , +15