Diethyl 1-fluoro-1-phenylsulfonylmethanephosphonate, a versatile agent for the preparation of monofluorinated building blocks.

Toru Koizumi, Toru Hagi, Yoshiharu Horie, Yoshio Takeuchi

Chemical and Pharmaceutical Bulletin · 1987 · 52 citations · 0 references

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Abstract

Diethyl 1-fluoro-1-phenylsulfonylmethanephosphonate was prepared and was transformed into 1-fluoroalkanephosphonate and phenyl 1-fluorovinyl sulfones, which are useful monofluorinated building blocks.