Synthesis of fluorine substituted pyrazolopyrimidines as potential leads for the development of PET-imaging agents for the GABAA receptors

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Atomic physicochemical parameters for three-dimensional-structure-directed quantitative structure-activity relationships. 2. Modeling dispersive and hydrophobic interactions

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Relationship between lipophilicity and brain extraction of C-11-labeled radiopharmaceuticals.

Michael J. Welch, Michael R. Kilbourn, Marcus E. Raichle · PubMed · 1983 · 286 citations

Pharmacy, Pharmacokinetics, Pharmacology +14

Imaging of [11C]-labelled RO 15-1788 binding to benzodiazepine receptors in the human brain by positron emission tomography

A. Persson, E. Ehrin, Lars I. Eriksson et al. · Journal of Psychiatric Research · 1985 · 174 citations

Medicine, Neuroscience, Pharmacology +13

[¹¹C]Flumazenil Positron Emission Tomography Visualizes Frontal Epileptogenic Regions

Ivanka Savić, J. O. Thorell, Per E. Roland · Epilepsia · 1995 · 132 citations

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