Expedient and Rapid Synthesis of 1,2,3-Triazolo[5,1-<i>c</i>]morpholines through Palladium−Copper Catalysis

Abstract

A one-pot approach using palladium-copper as catalyst has been developed for the synthesis of morpholines fused with 1,2,3-triazole. Good regioselectivity, mild reaction conditions, high yields and short reaction time are the hallmarks of this method.