Synthesis of 1,2,4-oxadiazole-linked orthogonally urethane-protected dipeptide mimetics

A general and expedient method for the solid-phase synthesis of 1,4-benzodiazepine derivatives

Barry A. Bunin, Jonathan A. Ellman · Journal of the American Chemical Society · 1992 · 444 citations

Combinatorial Chemistry, Derivative (Chemistry), 1,4-Benzodiazepine Derivatives +13

Bis(2-methoxyethyl)aminosulfur Trifluoride:  A New Broad-Spectrum Deoxofluorinating Agent with Enhanced Thermal Stability

G. S. LAL, Guido P. Pez, Reno J. Pesaresi et al. · The Journal of Organic Chemistry · 1999 · 394 citations

Halogenation, Organic Material Chemistry, Chemical Engineering +9

An Unnatural Biopolymer

Charles Y. Cho, Edmund J. Moran, Sara Cherry et al. · Science · 1993 · 361 citations

Medicinal Chemistry in the Golden Age of Biology: Lessons from Steroid and Peptide Research

Ralph Hirschmann · Angewandte Chemie International Edition in English · 1991 · 228 citations

Rational Drug Discovery, Drug Target, Quantitative Pharmacology +25

Design, Synthesis, and Evaluation of Phe-Gly Mimetics:  Heterocyclic Building Blocks for Pseudopeptides

Susanna Borg, Roeland C. Vollinga, Maryse Labarre et al. · Journal of Medicinal Chemistry · 1999 · 148 citations · Full text

Combinatorial Chemistry, Peptide Engineering, Organic Chemistry +16