Selective arylation of 2-substituted indoles towards 1,2- and 2,3-functional indoles directed through the catalytic system

A General and Efficient Copper Catalyst for the Amidation of Aryl Halides and the <i>N</i>-Arylation of Nitrogen Heterocycles

Artis Klapars, Jon C. Antilla, Xiaohua Huang et al. · Journal of the American Chemical Society · 2001 · 1K citations

Natural Sciences, Chemistry, Catalysis +11

Synthesis of indoles via palladium-catalyzed heteroannulation of internal alkynes

Richard C. Larock · Journal of the American Chemical Society · 1991 · 824 citations

Natural Sciences, Chemistry, Analytical Chemistry +11

Room-Temperature Palladium-Catalyzed Amination of Aryl Bromides and Chlorides and Extended Scope of Aromatic C−N Bond Formation with a Commercial Ligand

John F. Hartwig, Motoi Kawatsura, Sheila I. Hauck et al. · The Journal of Organic Chemistry · 1999 · 764 citations

Natural Sciences, Chemistry, Catalysis +9

Room Temperature Palladium-Catalyzed 2-Arylation of Indoles

Nicholas R. Deprez, Dipannita Kalyani, Andrew L. Krause et al. · Journal of the American Chemical Society · 2006 · 646 citations

Natural Sciences, Chemistry, Catalysis +15

Direct Palladium-Catalyzed C-2 and C-3 Arylation of Indoles:  A Mechanistic Rationale for Regioselectivity

Benjamin S. Lane, Meghann A. Brown, Dalibor Sameš · Journal of the American Chemical Society · 2005 · 645 citations

Natural Sciences, Chemistry, Medicinal Chemistry +16