Concepedia

Structure-activity relationship of a series of diaminoalkyl substituted benzimidazole as neuropeptide Y Y1 receptor antagonists

Hamideh Zarrinmayeh, Dennis M. Zimmerman, Buddy E. Cantrell, Douglas A. Schober, Robert E. Bruns, Susan L. Gackenheimer, Paul L. Ornstein, Philip A. Hipskind, Thomas C. Britton, Donald R. Gehlert

Bioorganic & Medicinal Chemistry Letters · 1999 · 91 citations · 16 references

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16

Neuropeptide Y—a novel brain peptide with structural similarities to peptide YY and pancreatic polypeptide

Kazuhiko Tatemoto, Mats Carlquist, Viktor Mutt · Nature · 1982 · 2.3K citations

, , +15

A receptor subtype involved in neuropeptide-Y-induced food intake

Christophe Gerald, Mary W. Walker, Leoluca Criscione et al. · Nature · 1996 · 893 citations

, , +14

Neuropeptide Y Stimulates Feeding but Inhibits Sexual Behavior in Rats*

John T. Clark, Pushpa S. Kalra, Satya P. Kalra · Endocrinology · 1985 · 393 citations

, , +17

The first highly potent and selective non-peptide neuropeptide Y Y1 receptor antagonist: BIBP3226

K Rudolf, Wolfgang Eberlein, Wolfhard Engel et al. · European Journal of Pharmacology · 1994 · 374 citations

, , +7

Evidence for neuropeptide Y mediation of eating produced by food deprivation and for a variant of the Y1 receptor mediating this peptide's effect

B. Glenn Stanley, William Magdalin, Alexander Seirafi et al. · Peptides · 1992 · 289 citations

, , +16