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Design, synthesis, and structure–activity relationship study of conformationally constrained analogs of indole-3-carboxamides as novel CB1 cannabinoid receptor agonists

Takao Kiyoi, Mark York, Stuart Francis, Darren Edwards, Glenn Walker, Andrea K. Houghton, Jean E. Cottney, James Α. Baker, Julia M. Adam

Bioorganic & Medicinal Chemistry Letters · 2010 · 17 citations · 6 references

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6

Allosteric Modulation of the Cannabinoid CB1 Receptor

M. R. Price, Gemma L. Baillie, Adèle Thomas et al. · Molecular Pharmacology · 2005 · 440 citations

Ring-substituted quinolines as potential anti-tuberculosis agents

Suryanarayana Vangapandu, Meenakshi Jain, Rahul Jain et al. · Bioorganic & Medicinal Chemistry · 2004 · 102 citations

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A role for cannabinoid receptors, but not endogenous opioids, in the antinociceptive activity of the CB2-selective agonist, GW405833

Garth T. Whiteside, Susan L. Gottshall, Jamie Boulet et al. · European Journal of Pharmacology · 2005 · 93 citations

, , +15

Reduction of quinolines to 1,2,3,4-tetrahydro derivatives employing a combination of NaCNBH3 and BF3.OEt2

A. Srikrishna, T. Jagadeeswar Reddy, R. Viswajanani · Tetrahedron · 1996 · 53 citations

, , +5

Design, synthesis, and structure–activity relationships of indole-3-carboxamides as novel water soluble cannabinoid CB1 receptor agonists

Julia M. Adam, Jim Cairns, Wilson Caulfield et al. · MedChemComm · 2010 · 36 citations

, , +17