Synthesis, stabilization and formulation of [177Lu]Lu-AMBA, a systemic radiotherapeutic agent for Gastrin Releasing Peptide receptor positive tumors

Synthesis and Evaluation of Bombesin Derivatives on the Basis of Pan-Bombesin Peptides Labeled with Indium-111, Lutetium-177, and Yttrium-90 for Targeting Bombesin Receptor-Expressing Tumors

Hanwen Zhang, Jianhua Chen, Christian Waldherr et al. · Cancer Research · 2004 · 197 citations

Medicinal Chemistry, Drug Target, Pan-bombesin Peptides +15

177Lu-AMBA: Synthesis and characterization of a selective 177Lu-labeled GRP-R agonist for systemic radiotherapy of prostate cancer.

Laura E. Lantry, Enrico Cappelletti, Mary Ellen Maddalena et al. · PubMed · 2006 · 175 citations

The addition of DTPA to [177Lu-DOTA0,Tyr3]octreotate prior to administration reduces rat skeleton uptake of radioactivity

Wouter A.P. Breeman, Katy van der Wansem, Bert F. Bernard et al. · European Journal of Nuclear Medicine and Molecular Imaging · 2003 · 73 citations

Positron Emission Tomography, Skeleton Uptake, Medicine +10

Development of an in vitro model for assessing the in vivo stability of lanthanide chelates

W.P Li, Dangshe Ma, C. Higginbotham et al. · Nuclear Medicine and Biology · 2001 · 67 citations

Pharmaceutical Science, Engineering, Medicine +8

Selenomethionine protects against adverse biological effects induced by space radiation

Ann R. Kennedy · Free Radical Biology and Medicine · 2004 · 67 citations

Health Sciences, Medicine, Radiation Effect +7