Microwave-assisted synthesis of some novel 1,2,3-triazoles by click chemistry, and their biological activity

A Stepwise Huisgen Cycloaddition Process: Copper(I)-Catalyzed Regioselective “Ligation” of Azides and Terminal Alkynes

Vsevolod V. Rostovtsev, Luke G. Green, Valery V. Fokin et al. · Angewandte Chemie International Edition · 2002 · 11.5K citations

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Synthesis and anticancer activity of chalcone-pyrrolobenzodiazepine conjugates linked via 1,2,3-triazole ring side-armed with alkane spacers

Ahmed Kamal, S. Prabhakar, M. Janaki Ramaiah et al. · European Journal of Medicinal Chemistry · 2011 · 145 citations

Pharmacy, Medicinal Chemistry, Pharmacology +14

Synthesis of 4‐aminoquinoline‐1,2,3‐triazole and 4‐aminoquinoline‐1,2,3‐triazole‐1,3,5‐triazine Hybrids as Potential Antimalarial Agents

Sunny Manohar, Shabana I. Khan, Diwan S. Rawat · Chemical Biology & Drug Design · 2011 · 116 citations

Pharmacy, Medicinal Chemistry, Pharmacology +12

Efficient synthesis and in vitro antitubercular activity of 1,2,3-triazoles as inhibitors of Mycobacterium tuberculosis

Poovan Shanmugavelan, Sangaraiah Nagarajan, Murugan Sathishkumar et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 105 citations

Pharmacy, Medicinal Chemistry, Pharmacology +13

Synthesis and structure–activity relationship of 1- and 2-substituted-1,2,3-triazole letrozole-based analogues as aromatase inhibitors

Jérémie A. Doiron, Al Halifa Soultan, Ryan Richard et al. · European Journal of Medicinal Chemistry · 2011 · 86 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13