Concepedia

9‐Phenanthrol inhibits human TRPM4 but not TRPM5 cationic channels

Teddy Grand, Marie Demion, Caroline Norez, Yvette Mettey, Pierre Launay, Frédéric Becq, P Bois, Romain Guinamard

British Journal of Pharmacology · 2008 · 156 citations · 30 references

DOIFull text

Open access

Abstract

We identify 9-phenanthrol as a TRPM4 inhibitor, without effects on TRPM5. It could be valuable in investigating the physiological functions of TRPM4, as distinct from those of TRPM5.

References

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